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2 404 185

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IPC

C07D498/02(2006-01-01)

C07D413/14(2006-01-01)

A61K31/42(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2009114406/04, 2009-04-16

(24)

Start date

2009-04-16

(22)

Actual filing date

2009-04-16

(45)

Published

2010-11-20

(72)

Inventor

Mjasoedov Nikolaj FedorovichShevchenko Valerij PavlovichNagaev Igor' JulianovichBobrov Mikhail Jur'EvichBezuglov Vladimir Vilenovich

(73)

Holder

Uchrezhdenie Rossijskoj Akademii Nauk Institut Molekuljarnoj Genetiki Ran Ran)

UNIFORMLY TRITIUM-LABELLED (R)-(+)-[5-METHYL-3-(4-MORPHOLINYLMETHYL) -2,3-DIHYDRO-[1,4]OXAZINE[2,3,4-hi]-6-INDOLYL]-1-NAPHTHALINYLMETHANONE ACETATE Russian patent published in 2010 - IPC C07D498/02 C07D413/14 A61K31/42 A61P29/00

Abstract RU 2404185 C1

FIELD: chemistry.

SUBSTANCE: invention relates to uniformly tritium-labelled (R)-(+)-[5-methyl-3-(4-morpholinylmethyl)-2,3-dihydro-[1,4]oxazine[2,3,4-hi]-6-indolyl]-1-naphthalinylmethanone acetate of formula I: .

EFFECT: wide range of labelled analogues of physiologically active compounds.

1 ex

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RU 2 404 185 C1

Authors

Mjasoedov Nikolaj Fedorovich

Shevchenko Valerij Pavlovich

Nagaev Igor' Julianovich

Bobrov Mikhail Jur'Evich

Bezuglov Vladimir Vilenovich

Dates

2010-11-20—Published

2009-04-16—Filed