FIELD: chemistry.
SUBSTANCE: present invention relates to novel heterocyclyl-pyrimidinyl-amino derivatives of formula (I), and agrochemically acceptable salts thereof, intermediate compounds of formula (II) for production thereof, fungicide compositions and a method of controlling phytopathogens and fungi, primarily of plants. In the compound of general formulae and , Het denotes a heterocycle selected from a group consisting of: , Y independently denotes a halogen atom, C1-C8-alkyl, C1-C8-haloalkyl with 1-5 halogen atoms, C1-C8-alkylamino, di-C1-C8-alkylamino, C1-C8-alkoxy, C1-C8-haloalkoxy with 1-5 halogen atoms, C2-C8-haloalkenyloxy with 1-5 halogen atoms, substituted with C1-C8-alkyl or unsubstituted C1-C8-alkoxyalkyl, substituted with C1-C8-alkyl or unsubstituted C1-C8-haloalkoxyalkyl with 1-5 halogen atoms; p equals 0, 1 or 2; Ra denotes a hydrogen atom, C1-C4-alkyl, C3-C6-cycloalkyl, C1-C4-haloalkyl with 1-5 halogen atoms; Rb and Rc independently denote a hydrogen atom, a halogen atom, C1-C4-alkyl, C1-C4-haloalkyl with 1-5 halogen atoms; X independently denotes C1-C4-alkyl, C1-C4-haloalkyl or a halogen atom; n equals 0, 1 or 2; L1 and L2 independently denote a hydrogen atom, C1-C8-alkyl, unsubstituted or substituted with C1-C8-alkoxy, di-C1-C8-alkylamino, hydroxy or C3-C6-cycloalkyl; C3-C6-cycloalkyl; C1-C4-haloalkyl with 1-5 halogen atoms; C3-C6-halocycloalkyl with 1-5 halogen atoms; C2-C6-alkenyl; C2-C6-alkynyl; C1-C4-alkoxy; C1-C4-haloalkoxy with 1-5 halogen atoms; C2-C6-alkenyloxy; C2-C6-alkynyloxy; C2-C6-haloalkenyloxy with 1-5 halogen atoms; C2-C6-haloalkynyloxy with 1-5 halogen atoms; (2-oxopyrrolidin-1-yl)- C1-C8-alkyl; (2-oxopyrrolidin-1-yl)-C1-C8-haloalkyl with 1-5 halogen atoms, W denotes a leaving group such as a halogen atom.
EFFECT: efficiency of the compound.
14 cl, 4 dwg, 128 ex
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Authors
Dates
2013-01-10—Published
2008-06-06—Filed