FIELD: organic chemistry. SUBSTANCE: product: 4-[2-(2-hydroxy-2-phenylethylamino)ethoxy]-phenylacetic acid of the formula 4-C6H5CH(OH)CH2NHCH2CH2OC6H4CH2COOH or its bioprecursor taken from amide or ester, or pharmaceutically acceptable salt and pharmaceutical composition. Reagent 1: styrene oxide. Reagent 2: 4-(H2NCH2CH2O)C6H4CH2COR4, COR4-amide group. Reaction conditions: at heating and at the following if necessary product hydrolysis to prepare acid and conversion of the latter if necessary to ester and product isolation if necessary as pharmaceutically acceptable salt. Synthesized compounds were used as bioactive substances and can be used in medicine. EFFECT: improved method of synthesis. 12 cl, 4 tbl
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