FIELD: organic chemistry, medicine, hematology, pharmacy.
SUBSTANCE: invention relates to novel compounds of the formula (I): in all their stereoisomeric forms and their mixtures taken in any ratio and their physiologically acceptable salts possessing properties of inhibitors of factor Xa and/or factor VIIa, and to a medicinal agent based on thereof. Also, invention relates to a method for synthesis of these compounds and their using for preparing pharmaceutical agents for inhibition of activity of factor Xa and/or factor VIIa or for their effect on blood coagulation or fibrinolysis.
EFFECT: valuable medicinal properties of compounds and pharmaceutical composition.
10 cl, 1 tbl, 276 ex
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Authors
Dates
2007-05-27—Published
2002-11-08—Filed