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(19)

RU

(11)

2 332 401

(13)

C2

(51)

IPC

C07D211/06(2006-01-01)

A61K31/4468(2006-01-01)

A61P25/06(2006-01-01)

A61P25/14(2006-01-01)

A61P25/16(2006-01-01)

A61P25/18(2006-01-01)

A61P25/24(2006-01-01)

A61P25/28(2006-01-01)

(21) (22)

Application

2005125918/04, 2004-01-15

(24)

Start date

2004-01-15

(22)

Actual filing date

2004-01-15

(45)

Published

2008-08-27

(72)

Inventor

Uehjner Dehvid M.Dehvis Robert E.Brehnn Mark R.

(73)

Holder

Akadia Farmas'Jutikalz Ink.

SELECTIVE SEROTONIN 2A/2C RECEPTOR INVERSE AGONISTS, USED AS THERAPEUTICS FOR NEURODEGENERATIVES DISEASES Russian patent published in 2008 - IPC C07D211/06 A61K31/4468 A61P25/06 A61P25/14 A61P25/16 A61P25/18 A61P25/24 A61P25/28 

Abstract RU 2332401 C2

FIELD: chemistry.

SUBSTANCE: invention relates to the compound with formula (I) or to its tartrate salt. The invention also relates to application of the composition as well as the method of inhibiting of monoamine receptor activation to inverse agonist and anti-dyskinesia agent in the combination with inverse agonist.

EFFECT: production of the new biologically active compound having inverse agonist activity of serotonin receptor.

54 cl, 7 ex, 3 tbl

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RU 2 332 401 C2

Authors

Uehjner Dehvid M.

Dehvis Robert E.

Brehnn Mark R.

Dates

2008-08-27—Published

2004-01-15—Filed

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