NEW COMPOUNDS AS MODULATOR OF OPIOTIC RECEPTORS Russian patent published in 2008 - IPC C07D401/04 A61K31/4439 A61K31/4725 A61P25/04 

Abstract RU 2332411 C2

FIELD: chemistry.

SUBSTANCE: invention relates to the compounds of general formula I , where: X denotes (CR15R16)m-, where: m is 1, R15 and R16- hydrogen; R1 selected from the group consisting of

A-B selected from the group consisting of N-C, C-N, N-N and C-C; D-E selected from the group consisting of O-C, S-C and O-N. The compounds can be used for the treatment of disorders modulated by opiotic receptors, for example, pain and gastroenteric disorder. The method of pharmaceutical composition production and application of the compounds are described.

EFFECT: production of the new compounds for the treatment of disorders modulated by opiotic receptors.

41 cl, 2 tbl, 18 ex

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RU 2 332 411 C2

Authors

Breslin Genri Dzh.

Khe Vej

Kavash Robert V.

Dates

2008-08-27Published

2003-04-17Filed