DIPYRAZOLES AS CENTRAL NERVOUS SYSTEM AGENTS Russian patent published in 2010 - IPC C07D231/22 C07D231/26 C07D401/14 A61K31/415 A61P25/08 A61P25/28

Abstract RU 2401258 C2

FIELD: chemistry.

SUBSTANCE: invention is aimed at dipyrazole compounds of formula I and their pharmaceutically acceptable salts, where radicals and groups are defined in claim 1 of the formula of invention. Disclosed compounds modulate AMPA and NMDA receptor functioning. A pharmaceutical composition based on formula I compounds and separate dipyrazole compounds are also part of the subject of invention.

EFFECT: possibility of using compounds as pharmaceutical agents, mainly for treating psychoneurological diseases.

16 cl, 2 tbl, 39 ex

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RU 2 401 258 C2

Authors

Kosli Rehjmond V. Ml.

Makdonald Duglas

Sher Rouzi

Dates

2010-10-10—Published

2006-03-15—Filed