NEUROTROPIC DRUG AND METHOD FOR ITS PRODUCTION Russian patent published in 2009 - IPC C07D213/82 A61K31/455 A61P25/28

Abstract RU 2359962 C1

FIELD: chemistry.

SUBSTANCE: invention is related to new compound - 1-((3-pyridylcarbonyl)aminomethyl)-1-cyclohexane acetic acid of formula I and its pharmaceutically acceptable salts, which display nootropic, anticonvulsive, anxiolytic properties and may find application as neurotropic drug. Compound I is produced by condensation of alkyl ether of 3-pyridine-carbonic acid with salt 1-(aminomethyl)cyclohexane acetic acid, normally, in organic dissolvent at dissolvent boiling temperature with further treatment with mineral or organic acid, if required.

EFFECT: in order to produce salt of compound I, it is treated usually with oxide hydrate or oxide of alkaline or alkali-earth metal.

5 cl, 8 tbl, 5 ex

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RU 2 359 962 C1

Authors

Kopelevich Vjacheslav Mikhajlovich

Pozdnev Vladimir Fedorovich

Dates

2009-06-27—Published

2007-12-13—Filed