17,17-DIMETHYL-D-HOMO-B-NOR-8α-OESTRONE HAVING HYPOLIPIDEMIC AND CARDIOPROTECTOR ACTIVITY Russian patent published in 2010 - IPC C07J63/00 A61P3/06 

Abstract RU 2391351 C1

FIELD: chemistry.

SUBSTANCE: invention relates to biologically active analogues of steroid oestrogens. 17,17-dimethyl-D-homo-B-nor-8α-oestrone is synthesised, which has noticeably pronounced hypolipidemic and cardioprotector activity in the absence of uterotropic action. 17,17-dimethyl-D-homo-B-nor-8α-oestrone.

EFFECT: obtaining compounds which can be used in medicine as a basis for designing effective medicinal preparations for treating cardiovascular diseases.

1 cl, 1 ex, 4 tbl

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RU 2 391 351 C1

Authors

Shavva Aleksandr Grigor'Evich

Morozkina Svetlana Nikolaevna

Antimonova Ol'Ga Igorevna

Surinov Boris Pavlovich

Dates

2010-06-10Published

2008-12-25Filed