FIELD: chemistry.
SUBSTANCE: invention relates to a method of producing oxazoles of formula IV through condensation of aromatic aldehydes with α-ketoximes with formation of the corresponding N-oxides and their subsequent reaction with sulphonyl or thionyl compounds, preferably with inorganic thionyl halides or organic sulphonyl halides.
EFFECT: method is characterised by high output and purity of the obtained product, as well as avoiding the need to extract unstable intermediate N-oxides in form of individual compounds.
12 cl, 8 ex
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Authors
Dates
2010-10-27—Published
2005-12-01—Filed