COMPOUND, POSSESSING DETRUSOR-CONTRACTING AND URETHRAL SPHINCTER-RELAXING ACTIVITY Russian patent published in 2014 - IPC C07D277/20 C07D277/56 A61K31/426 A61P13/02 A61P13/10 A61K45/00 

FIELD: chemistry.

SUBSTANCE: invention relates to a compound, represented by formula (I) where represents α-configuration; represents β-configuration; and represents α-configuration, β-configuration or their arbitrary mixture, its salt, or its mixture with diastereomer in an arbitrary ratio, or its cyclodextrin clathrate. The invention relates to a pharmaceutical composition for the prevention, treatment and/or reduction of intensity of the urinary bladder contraction dysfunction and/or urethral relaxation dysfunction, which contains the compound, represented by formula (I) as an active ingredient. The invention also relates to a compound, represented by formula (I-a) where R¹ represents C₁-C₄-alkyl group, such as methyl, ethyl, propyl, isopropyl, butyl, isobutyl or tert-butyl; represents α-configuration; represents β-configuration; and represents α-configuration, β-configuration or their arbitrary mixture, its salt, or its mixture with diastereomer in an arbitrary ratio, or its cyclodextrin clathrate.

EFFECT: compound in accordance with the claimed invention is suitable as an excellent agent for the prevention, treatment and/or improvement of the insufficiently active urinary bladder.

8 cl, 3 tbl, 8 dwg, 24 ex