AMINE SALT AND CRYSTALS THEREOF Russian patent published in 2018 - IPC C07D277/20 C07D277/56 C07D211/22 C08B37/16 A61K31/426 A61K47/40 A61P13/02 A61P13/10 A61P43/00 

Abstract RU 2658823 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to a salt of a compound represented by the formula (I), where represents α-configuration, represents β-configuration and represents α-configuration, β-configuration or a mixture thereof in an arbitrary ratio, and 4-piperidinemethanol; a crystal thereof; or cyclodextrin clathrate thereof. Compound of the invention can be represented by general formula (II). (I), (II).

EFFECT: compound is an agent for reducing bladder detrusor and relaxation of the urethral sphincter, and also for prevention, treatment and/or alleviation of a hypoactive bladder.

23 cl, 6 tbl, 20 ex

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RU 2 658 823 C2

Authors

Tani Kousuke

Kinosita Akikhiro

Khanada Kejsuke

Aratani Esiyuki

Nekado Takakhiro

Simabukuro Atsusi

Dates

2018-06-25Published

2013-08-30Filed