WATER-SOLUBLE SALAMIDE DERIVATIVE POSSESSING TRANQUILISING, NOOTROPIC AND ANALGESIC ACTIVITY Russian patent published in 2015 - IPC A61K31/625 A61P25/22 A61P25/28 A61P29/00 

Abstract RU 2540464 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention can be used in chemical-pharmaceutical industry for preparing effective tranquilising salamide preparations and analgesics. What is presented is using salicyloyl morpholine sodium salt of formula (I) as a tranquilising, nootropic and analgesic agent possessing low gastric toxicity.

EFFECT: implementing the declared application with the therapeutic index of salicyloyl morpholine of formula (I) is 3 times higher than that of mexidole, and 9,5 times higher than that of aspirin.

5 tbl

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RU 2 540 464 C2

Authors

Brel' Anatolij Kuz'Mich

Petrov Vladimir Ivanovich

Lisina Svetlana Viktorovna

Kovalev Dmitrij Gennad'Evich

Salomatina Julija Nikolaevna

Mjagkova Irina Alekseevna

Dates

2015-02-10Published

2012-05-28Filed