SOLID COMPOSITIONS CONTAINING AGONIST TO GLP AND SALT OF N-(2-HYDROXYBENZOYL)AMINO)CAPRYLIC ACID Russian patent published in 2016 - IPC A61K38/26 A61K9/20 A61P3/10 

Abstract RU 2600440 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: group of inventions concerns solid compositions containing agonist GLP-1 and salt of N-(8-(2-hydroxybenzoyl)amino)caprylic acid, where the amount of said salt is at least 0.6 or at least 0.8 mmol, and said GLP-1 agonist represents semaglutide, as well as use in medicine for treating type II diabetes or obesity.

EFFECT: group of inventions provides improved action and bioavailability.

28 cl, 1 ex, 10 tbl

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RU 2 600 440 C2

Authors

Zauerberg Per

Berregaard Simon

Nilsen Flemming Sajer

Dates

2016-10-20Published

2011-12-16Filed