POTENT COMPSTATIN ANALOGS Russian patent published in 2018 - IPC C07K7/08 A61K38/10 A61P37/00 

Abstract RU 2656102 C2

FIELD: chemistry.

SUBSTANCE: suggested method of preparing a compound that inhibits the activation of complement, where the said compound is Xaa1-Cys-Val-Xaa2-Gln-Asp-Xaa3-Gly-Xaa4-His-Arg-Cys-Xaa5 (SEQ ID NO:26).

EFFECT: given compounds show significantly higher activity in inhibiting complement activation in comparison with the currently available compounds.

22 cl, 6 tbl, 8 dwg, 11 ex

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RU 2 656 102 C2

Authors

Lembriz Dzhon D.

Katragadda Madan

Dates

2018-05-31Published

2012-11-06Filed