(HETERO)ARYL CYCLOPROPYLAMINE COMPOUNDS AS LSD1 INHIBITORS Russian patent published in 2019 - IPC C07D205/04 C07D207/14 C07D209/96 C07D211/56 C07D215/38 C07D221/20 C07D223/12 C07D309/14 C07D401/12 C07D405/12 A61K31/44 A61P35/02 

Abstract RU 2681211 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds of formula I, as well as use thereof in the treatment or prevention of cancer or viral infection associated with LSD1.

I.

EFFECT: obtaining novel compounds (hetero)aryl cyclopropylamines having inhibitory activity of lysine-specific demethylase-1 (LSD1).

77 cl, 3 tbl

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RU 2 681 211 C2

Authors

Ortega-Munos Alberto

Fajf Mattyu Kolin Tor

Martinell-Pedemonte Mark

Estyarte-Martines Mariya-De-Los-Ankheles

Valls-Vidal Nuriya

Kurts Guido

Kastro-Palomino-Lariya Khulio-Sesar

Dates

2019-03-05Published

2012-10-22Filed