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2 750 488

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IPC

C07J43/00(2006-01-01)

A61K31/58(2006-01-01)

A61P13/08(2006-01-01)

A61P3/00(2006-01-01)

A61P29/00(2006-01-01)

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Application

2020118189, 2020-06-03

(24)

Start date

2020-06-03

(22)

Actual filing date

2020-06-03

(45)

Published

2021-06-28

(72)

Inventor

Sorokina Irina VasilevnaPopadyuk Irina IgorevnaZhukova Natalya AnatolevnaNizomov Sirozhiddin AshuralievichMeshkova Yuliya VladimirovnaBaev Dmitrij SergeevichBorisov Sergej AlkisovichSalomatina Oksana VladimirovnaTolstikova Tatyana GenrikhovnaSalakhutdinov Nariman Faridovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Novosibirskij Institut Organicheskoj Khimii Im. N.N. Vorozhtsova Sibirskogo Otdeleniya Rossijskoj Akademii Nauk So Ran)

1,2,4-OXADIAZOLE DERIVATIVES OF DESOXYCHOLIC ACID, EXHIBITING PROSTATE-PROTECTIVE EFFECT, HYPOCHOLESTEROLEMIC AND ANTI-INFLAMMATORY ACTIVITY Russian patent published in 2021 - IPC C07J43/00 A61K31/58 A61P13/08 A61P3/00 A61P29/00

Abstract RU 2750488 C1

FIELD: chemistry.

SUBSTANCE: invention relates to pharmaceutical chemistry, specifically to compounds constituting oxadiazole derivatives of deoxycholic acid by the formula I, wherein R constitutes Me or Ph.

EFFECT: technical result consists in expanding the range of prostatoprotective substances also exhibiting pleiotropic - anti-inflammatory and hypocholesterolemic effects.

1 cl

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RU 2 750 488 C1

Authors

Sorokina Irina Vasilevna

Popadyuk Irina Igorevna

Zhukova Natalya Anatolevna

Nizomov Sirozhiddin Ashuralievich

Meshkova Yuliya Vladimirovna

Baev Dmitrij Sergeevich

Borisov Sergej Alkisovich

Salomatina Oksana Vladimirovna

Tolstikova Tatyana Genrikhovna

Salakhutdinov Nariman Faridovich

Dates

2021-06-28—Published

2020-06-03—Filed