FIELD: biotechnology.
SUBSTANCE: present invention relates to the field of biotechnology, specifically to a new conjugate of a stabilized agonist of a glucagon-like peptide-1 (GLP-1) receptor; it can be used in medicine. The invention allows for producing the conjugate with improved pharmacological properties: delayed release balances the agonist stability with the speed of release in the organism environment, providing its longer action in comparison with known analogues.
EFFECT: invention can be used in medicinal practice, when treating patients suffering from diabetes or other similar metabolic disorders, using schemes including the administration of a dose once a month or less.
16 cl, 16 dwg, 2 tbl, 8 ex
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Authors
Dates
2022-01-18—Published
2017-03-16—Filed