(2S,4S)-4-AMINO-N-(4-FLUOROPHENYL)PYROGLUTAMIC ACID EXHIBITING CEREBROPROTECTIVE, NOOTROPIC, AND ANTITHROMBOTIC ACTION Russian patent published in 2022 - IPC C07D207/28 A61K31/4015 A61P25/28 

Abstract RU 2769521 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a new derivative of pyroglutamic acid - (2S,4S)-4-amino-N-(4-fluorophenyl)pyroglutamic acid by the formula 1.

EFFECT: production of a new compound applicable as a cerebral protector with nootropic and antithrombotic activity.

1 cl, 6 tbl, 7 ex

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RU 2 769 521 C1

Authors

Charushin Valerij Nikolaevich

Vigorov Aleksej Yurevich

Krasnov Viktor Pavlovich

Nizova Irina Albertovna

Matveeva Tatyana Viktorovna

Levit Galina Lvovna

Tyurenkov Ivan Nikolaevich

Bakulin Dmitrij Aleksandrovich

Kovalev Nikolaj Sergeevich

Kurkin Denis Vladimirovich

Nazarov Oleg Igorevich

Dates

2022-04-01Published

2021-02-17Filed