A-EXO-AZASPIRO-INHIBITORS OF THE MENIN-MLL INTERACTION Russian patent published in 2023 - IPC C07D495/04 C07D519/00 A61P35/02 A61P3/10 

Abstract RU 2795096 C2

FIELD: medicinal chemistry.

SUBSTANCE: new compounds of formula (I), where the values of A, L, Y1, Y2, R1-R3, n1, n2, m1, m2 are defined in the claims, to a pharmaceutical composition containing such compounds, and to their use as inhibitors of menin-MLL protein-protein interactions.

EFFECT: useful in the treatment of diseases such as cancer, myelodysplastic syndrome (MDS) and diabetes.

10 cl, 4 tbl, 198 ex

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RU 2 795 096 C2

Authors

Daj, Syuedun

Keroll, Olive Aleksis Zhorzh

Kroski, Deniel Dzhejson

Tsaj, Vej

Fu, Litsyan

Kun, Linlun

Lyu, Intao

Van, Chzhao-Kuj

Morshkhojzer Geb. Kherkert, Barbara

Pande, Vinet

Edvards, Dzhejms Patrik

Patrik, Aaron Nataniel

Anzhibo, Patrik Rene

Ponsele, Virzhini Sofi

Dates

2023-04-28Published

2018-12-19Filed