FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes imidazodiazepines of the general formula (I) 
where values A, Q, R1, R2, R3, R4 are given in p. 1 of the invention claim. Compounds show the strong expressed anxiolytic, anticonvulsant, muscle relaxant and sedative-hypnotic properties. They form good water-soluble acid-additive salts and therefore can be used for preparing aqueous solutions for injection of drugs based on compounds of the formula (I) effectively. Invention describes also a method of synthesis of the above indicated compounds. EFFECT: improved method of synthesis, valuable pharmacological properties. 27 cl, 1 tbl, 259 ex
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