FIELD: organic chemistry. SUBSTANCE: invention relates to tricyclic derivatives of pyrazole of the general formula (I) where R1-R4 mean hydrogen, halogen atom, lower alkyl of lower alkoxy-group; R5 means lower alkyl; R6 means hydrogen atom, lower alkyl or lower alkoxy-group; X means -(CR7R8)n- or -CH=CH-; R7 and R8 mean hydrogen atom or lower alkyl and n = 1 or 2 or to pharmaceutically acceptable salts of basic compounds of the general formula (I). Compounds show ability to bind with serotonin-receptors and can be used for treatment or prophylaxis of central nervous system diseases, in part, for treatment of patients with sexual disorders and other diseases. Invention proposes also drug based on compounds of the formula (I) binding serotonin receptors and designated for treatment of sexual disorders. EFFECT: valuable medicinal and pharmacological properties of compounds. 12 cl, 3 dwg
Authors
Dates
2000-07-10—Published
1995-08-08—Filed