FIELD: medicine. SUBSTANCE: described are tricyclic benzazepine derivatives of general formula I: wherein Y,A,B,Z, R1, R2 are as defined in claims and method of preparing said derivatives, pharmaceutical composition based thereon, and method of inhibition of vasopressin. Invention is useful in treating states when it is desirable to reduce vasopressin levels such as cardial insufficiency, or the like. EFFECT: improved properties of the title compounds, and more efficient method of inhibition of vasopressin. 15 cl, 576 ex, 5 tbl
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