FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to novel 4-aryl-1- phenylalkyl-1,2,3,6-tetrahydropyridines of the formula (I) where Y is CH or -N-; R1 is H, halogen, CF3; R2 is H, halogen, (C3-C4)-alkyl or (C1-C4)-alkoxy-group; R3 and R4 means H or (C1-C3)-alkyl; X means: a) (C3-C6)-alkyl, (C3-C6)-alkoxy-group or (C1-C4)-alkoxycarbonyl-(C3-C6)-alkoxy-group; b) (C3-C7)-cycloalkyl or c) substitute taken among the group including phenyl, phenoxy, benzyl, their salts, solvates or quaternary ammonium salts. Compounds of the formula (I) show neurotropic and neuro- -protective activity and can be used in medicine for treatment of patients with central nervous system diseases. Invention relates to also intermediate compounds of the formula where is halogen atom or CF3 and formula (i) where R1, R2, R3, R4 and Y have values indicated for compounds of the formula (I) and W means methylene or carbonyl group. EFFECT: improved method of synthesis, valuable medicinal properties. 11 cl, 1 tbl, 39 ex
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