BENZOTHIENO[3,2-C]PYRIDINES, METHOD FOR THEIR PREPARING (VARIANTS), PHARMACEUTICAL COMPOSITION AND METHOD FOR ITS PREPARING Russian patent published in 2004 - IPC

Abstract RU 2222542 C2

FIELD: organic chemistry, chemical technology, pharmacy. SUBSTANCE: invention relates to benzothieno[3,2-c] pyridines of the formula (I) , their oxides, pharmaceutically acceptable additive salts and stereochemically isomeric forms wherein each R¹ represents independently hydrogen, halogen atom, C_1-6-alkyl or C_1-4-alkoxy-group; Alk represents C_1-6-alkanediyl; n = 1 or 2; p = 0, 1 or 2; D represents optionally substituted mono-, bi- or tricyclic nitrogen-containing heterocycle. These compounds elicit antagonistic activity with respect to central α2-adrenoceptors. Invention relates also to method for preparing compounds, compositions containing thereof and their using as medicinal preparations. EFFECT: improved preparing method, valuable medicinal properties of compounds. 13 cl, 2 tbl, 9 ex

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RU 2 222 542 C2

Authors

Kennis Ljudo Ehdmon Zhozefin

Piters Serzh Marija Aloisius

Bishoff Fransua Pol'

Dates

2004-01-27—Published

1999-10-01—Filed