CRYSTALLINE FORMS OF DERIVATIVE OF PYRIMIDINE NUCLEOSIDE (VARIANTS), PHARMACEUTICAL COMPOSITION, METHOD FOR PROPHYLAXIS AND TREATMENT OF TUMOR DISEASE AND APPLYING CRYSTALLINE FORM Russian patent published in 2005 - IPC

Abstract RU 2256666 C2

FIELD: organic chemistry, medicine, oncology, pharmacy.

SUBSTANCE: invention relates to new stable crystalline forms of derivative of pyrimidine nucleoside of the formula (I) eliciting the excellent anti-tumor activity. Also, invention relates to pharmaceutical composition eliciting an anti-tumor effect, applying crystalline form for preparing medicinal agent and to a method for prophylaxis or treatment of tumor diseases.

EFFECT: improved method for prophylaxis and treatment, valuable medicinal properties of derivative.

10 cl, 2 tbl, 4 dwg, 9 ex

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RU 2 256 666 C2

Authors

Takita Takasi

Okhtsuka Keiiti

Numagami Eidzi

Kharasima Susumu

Dates

2005-07-20Published

2002-02-06Filed