FIELD: medicine.
SUBSTANCE: method involves introducing 4-(4-methylpiperazine-1-ylmethyl)-N-[4-methyl-3-(4-pyridine-3-yl)pyrimidine-2-ylamino)phenyl]benzamide of formula I or its pharmaceutically permissible salt for preparing pharmaceutical compositions for treating CD117-positive non-operable and/or metastatic malignant gastrointestinal stromal tumors.
EFFECT: enhanced effectiveness of treatment.
6 cl, 1 tbl
Title | Year | Author | Number |
---|---|---|---|
TREATMENT OF PROLIFERATIVE ARTHRITIS | 2003 |
|
RU2322238C2 |
COMBINATION OF PYRIMIDYLAMINOBENZAMIDE AND IMANITIB DERIVATIVES FOR TREATMENT OR PREVENTION OF PROLIFERATIVE DISEASES | 2006 |
|
RU2430727C2 |
AMIDE DERIVATIVE, PHARMACEUTICAL COMPOSITION AND THERAPEUTIC AGENTS BASED ON THEREOF | 2003 |
|
RU2315043C2 |
COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS | 2006 |
|
RU2383545C2 |
USING DERIVATIVES OF N-PHENYL-2-PYRIMIDINEAMINE AGAINST MASTOCYTE-BASE DISEASES SIMILAR TO ALLERGIC DISTURBANCE | 2002 |
|
RU2304436C2 |
NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHIBITION OF TYROSINE KINASE ACTIVITY | 2011 |
|
RU2598852C2 |
NEW ANTHRANILAMIDOPYRIDINEUREAS AS VEGF RECEPTOR KINASE INHIBITORS | 2005 |
|
RU2415850C2 |
PHARMACEUTICAL COMPOSITION OF IMATINIB OR ITS PHARMACEUTICALLY ACCEPTABLE SALT, METHOD FOR PREPARING IT AND METHOD(S) OF TREATING | 2012 |
|
RU2517216C2 |
TRIAZOLOPYRIDINE JAK INHIBITOR COMPOUNDS AND METHODS | 2009 |
|
RU2561104C2 |
THERAPY OF TUMOURS WITH APPLICATION OF ANTIBODY TO VASCULAR ENDOTHELIAL GROWTH FACTOR AND ANTIBODIES TO HUMAN EPITHELIAL GROWTH FACTOR RECEPTOR TYPE 2 | 2007 |
|
RU2538664C2 |
Authors
Dates
2007-06-20—Published
2001-10-26—Filed