METHOD FOR PRODUCTION OF BETULINIC ACID Russian patent published in 2007 - IPC C07J53/00 C07J63/00 

Abstract RU 2305106 C1

FIELD: pharmaceutical industry, in particular production of anti-tumor and anti-HIV agents.

SUBSTANCE: claimed method includes reduction of betulonic acid with sodium borohydride in mixture of water and benzene in presence of phase transfer catalyst such as quaternary ammonium salt for 2 hours.

EFFECT: more effective method; increased yield of target product; decreased sodium borohydride consumption.

2 cl, 4 ex

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RU 2 305 106 C1

Authors

Kogaj Tamara Ivanovna

Kuznetsov Boris Nikolaevich

Dates

2007-08-27Published

2006-04-03Filed