COMBINATION OF SPECIFIC OPIOIDS WITH MUSCARINE ANTAGONISTS FOR INCONTINENCE THERAPY Russian patent published in 2007 - IPC A61K45/06 A61K31/135 A61K31/485 A61K31/46 A61P13/10 

Abstract RU 2305562 C2

FIELD: pharmaceutical chemistry and urology.

SUBSTANCE: invention proposes treatment of frequent vesical tenesmus and incontinence with combination of tramadol, its derivatives, and derivatives of 1-phenyl-3-dimethylaminopropane compounds of formula I: with antimuscarine agents, in particular combination of (+)-(2R,3R)-1-dimethylamino-3-(3-methoxyphenyl)-2-methylpentane-3-ol and oxybutynine. Invention also relates to drug form of this combination.

EFFECT: enlarged choice of incontinence treatment agents.

2 cl, 1 tbl, 2 ex

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RU 2 305 562 C2

Authors

Kristof Tomas

Dates

2007-09-10Published

2002-09-18Filed