Patenton — panteon of patents

(19)

RU

(11)

2 314 303

(13)

C2

(51)

IPC

C07D401/12(2006-01-01)

C07D417/12(2006-01-01)

C07D487/04(2006-01-01)

C07D495/04(2006-01-01)

C07D498/04(2006-01-01)

C07D513/04(2006-01-01)

A61K31/428(2006-01-01)

A61P7/02(2006-01-01)

A61P9/10(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2004106625/04, 2002-08-08

(24)

Start date

2002-08-08

(22)

Actual filing date

2002-08-08

(45)

Published

2008-01-10

(72)

Inventor

Okhta TosikharuKomorija SatosiJosino TosikharuUoto KouitiNakamoto JumiNaito KhirojukiMotizuki AkijosiNagata TsutomuKanno KhidejukiKhaginoja NorijasuJosikava KendziNagamoti MasatosiKobajasi SiozoOno Makoto

(73)

Holder

Dajiti Farmas'Jutikal Ko., Ltd.

DIAMINE DERIVATIVES Russian patent published in 2008 - IPC C07D401/12 C07D417/12 C07D487/04 C07D495/04 C07D498/04 C07D513/04 A61K31/428 A61P7/02 A61P9/10 A61P29/00 

Abstract RU 2314303 C2

FIELD: organic chemistry, medicine, hematology.

SUBSTANCE: invention relates to novel compounds or their salts that inhibit blood coagulation activated factor X and elicit strong anti-coagulating effect. Compounds are represented by one of the following formulae: Also, invention relates to a medicinal agent, inhibitor of blood coagulation activated factor X, anti-coagulating agent, medicinal composition comprising indicated compounds, to their using for preparing a medicinal agent, inhibitors and anti-coagulating agent.

EFFECT: valuable medicinal properties of compounds.

9 cl, 1 tbl, 794 ex

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RU 2 314 303 C2

Authors

Okhta Tosikharu

Komorija Satosi

Josino Tosikharu

Uoto Kouiti

Nakamoto Jumi

Naito Khirojuki

Motizuki Akijosi

Nagata Tsutomu

Kanno Khidejuki

Khaginoja Norijasu

Josikava Kendzi

Nagamoti Masatosi

Kobajasi Siozo

Ono Makoto

Dates

2008-01-10—Published

2002-08-08—Filed

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