METHOD FOR PREPARING 3β-ACETOXY-2-OXONORTARAXASTANE Russian patent published in 2008 - IPC C07J53/00 C07J63/00 

Abstract RU 2316561 C1

FIELD: organic chemistry, natural compounds, chemical technology, medicine.

SUBSTANCE: invention relates to a novel method for synthesis of 3β-acetoxy-20-oxonortaraxastane. Method involves interaction of chloroform extract prepared from plant Scotch thistle (Onopordum acanthium L.) flower receptacles comprising 3β-acetoxy-20-methylenetaraxastane with ozone excess in the mole ratio 3β-acetoxy-20-methylenetaraxastane : ozone = 1:1.5 at room temperature and stirring. The yield of the end product is 40%. Compound can be used as an antitumor and anti-inflammatory agent.

EFFECT: improved method of synthesis.

2 cl, 1 ex

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RU 2 316 561 C1

Authors

Akhmetova Vnira Rakhimovna

Shakurova Ehl'Vira Rifovna

Khalilova Alija Zufarovna

Khalilov Leonard Mukhibovich

Dates

2008-02-10Published

2006-04-24Filed