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2 739 559

(13)

(51)

IPC

C07J63/00(2006-01-01)

A61K31/56(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2020125244, 2020-07-30

(24)

Start date

2020-07-30

(22)

Actual filing date

2020-07-30

(45)

Published

2020-12-25

(72)

Inventor

Popov Sergei AleksandrovichSemenova Mariia DmitrievnaShults Elvira EduardovnaFrolova Tatiana Sergeevna

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Uchrezhdenie Nauki Novosibirskii Institut Organicheskoi Khimii Im. N.N. Vorozhtsova Sibirskogo Otdeleniia Rossiiskoi Akademii Nauk So Ran)

((3Β-ACETOXY-URS-12-EN-28-OYL-OXYACETOXY)METHYL)-1H-1,2,3-TRIAZOL-1-YL)METHYL)-4-METHYL-1,2,5-OXADIAZOL-2-OXIDE, HAVING SELECTIVE ANTICANCER ACTIVITY AGAINST MCF-7 BREAST CANCER CELLS Russian patent published in 2020 - IPC C07J63/00 A61K31/56 A61P35/00

Abstract RU 2739559 C1

FIELD: chemistry.

SUBSTANCE: invention relates to compound ((3β-acetoxy-urs-12-en-28-oyl-oxyacetoxy)methyl)-1H-1,2,3-triazol-1-yl)methyl)-4-methyl-1,2,5-oxadiazole-2-oxide.

EFFECT: obtaining a novel compound of formula 1, having selective anticancer activity on breast cancer cells MCF-7, which can find application in medicine.

1 cl, 1 tbl, 5 ex

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RU 2 739 559 C1

Authors

Popov Sergei Aleksandrovich

Semenova Mariia Dmitrievna

Shults Elvira Eduardovna

Frolova Tatiana Sergeevna

Dates

2020-12-25—Published

2020-07-30—Filed