PYRROLIDINE AND PIPERIDINE DERIVATIVES Russian patent published in 2008 - IPC C07D491/107 C07D207/14 C07D207/26 C07D207/50 C07D211/28 C07D211/30 C07D211/32 C07D211/34 C07D211/42 C07D211/56 C07D211/60 C07D211/72 C07D211/76 C07D401/04 C07D401/12 C07D401/14 C07D403/04 C07D413/12 C07D471/10 C07D487/10 C07D491/10 C07D498/10 C07D513/10 A61P1/00 A61P3/04 A61P3/10 A61P9/10 A61P11/00 A61P13/10 A61P15/00 A61P17/00 A61P25/00 A61P27/02 A61P29/00 A61P31/18 

Abstract RU 2326120 C9

FIELD: chemistry.

SUBSTANCE: invention pertains to new compound derivatives of pyrrolidine or piperidine with general formula (I) or their pharmaceutically acceptable salts: , where Ar1, Ar2, X1, R1, R2, R3, R4 , R5, R6, R7, R18, R32, R33, n2 are defined in the formula of invention.

EFFECT: compounds are antagonist to NK1.

24 cl, 113 ex

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RU 2 326 120 C9

Authors

Pelivol Sanil

Rejchard Gregori A.

Uong Cheng

Ksiao Dong

Tsui Khon-Chung

Shi Neng-Jang

Ehrridondo Khuan D.

Vrobleski Mishell' Lasi

Peleni Ehnenden

Dates

2008-06-10Published

2002-12-17Filed