FIELD: chemistry.
SUBSTANCE: description is given of a lactam-containing compound-derivative of tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide with formula I
, its pharmaceutical salt and pharmaceutical compositions, their content, and their use as Xa factor inhibitors. The given compound can be used for treating thromboembolic diseases.
EFFECT: obtaining a lactam-containing compound, which can be used for treating thromobembolic diseases.
42 cl, 9 tbl, 140 ex
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Authors
Dates
2009-02-10—Published
2002-09-17—Filed