LACTAM-CONTAINING COMPOUND AND ITS DERIVATIVES AS Xa FACTOR INHIBITORS Russian patent published in 2009 - IPC C07D471/04 A61K31/437 A61P7/02 

Abstract RU 2345993 C2

FIELD: chemistry.

SUBSTANCE: description is given of a lactam-containing compound-derivative of tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide with formula I , its pharmaceutical salt and pharmaceutical compositions, their content, and their use as Xa factor inhibitors. The given compound can be used for treating thromboembolic diseases.

EFFECT: obtaining a lactam-containing compound, which can be used for treating thromobembolic diseases.

42 cl, 9 tbl, 140 ex

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RU 2 345 993 C2

Authors

Pinto Donald

Kvan Mimi

Orueht Majkl

Li Jun-Long

Khan Vej

Kiao Dzhennifer

Lehm Patrik

Koch Stefani

Dates

2009-02-10Published

2002-09-17Filed