ENHANCED FINISHED FORMULATIONS CONTAINING SUBSTITUTED IMIDASOL DERIVATIVES Russian patent published in 2009 - IPC A61K9/22 A61K31/417 

Abstract RU 2349305 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention concerns medicines and quick dispersed solid dosaged formulation including effective dosage of substituted imidasol derivative as active component, of the general formula (I), where each of R1, R2, R3 and Y is as indicated in claim, or in the form of pharmaceutically acceptable salt, such as acid-added salt, e.g. hydrochloride, compounds of the general formula (I) featuring grid structure of active component and water soluble or dispersible carrier inert towards the active component. The grid structure is obtained by solvent sublimation from solid composition including active component and carrier solution in the solvent, facilitating pre-gastric absorption of active component.

EFFECT: improved imidasol derivative delivery.

17 cl, 4 tbl, 8 ex

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RU 2 349 305 C2

Authors

Behnberi S'Juzi

Jujarvi Paivi

Groter Leon P.

Lansmehnn Uolter

Mjurrej Ouehn

Savola Jukha-Matti

Dates

2009-03-20Published

2003-11-03Filed