DERIVATIVES OF IMIDAZO-PYRIDINE, WITH AFFINITY TO MELANOCORTIN RECEPTOR Russian patent published in 2009 - IPC C07D471/04 A61K31/4188 A61K31/4353 A61P25/04 A61P25/24 

Abstract RU 2358974 C2

FIELD: chemistry.

SUBSTANCE: described are new derivatives of imidazo-pyridine with general formula I in racemic, enantiomeric form or in combination of these forms, and their pharmaceutically used salts. Radicals R1-R4 are described in the description.

EFFECT: these compounds have affinity to melanocortin receptor; possibility of using them in making medicinal agents for treating disorders, related to body weight, mental disorders, pain, sexual activity disorders.

21 cl, 5 ex, 1 tbl

Similar patents RU2358974C2

Title Year Author Number
NEW DERIVATIVES BENZIMIDAZOLE AND IMIDAZOPYRIDINE AND THEIR APPLICATION AS MEDICINES 2004
  • Puatu Lidi
  • Bro Valeri
  • Sakjur Karol'
  • Ruber P'Er
  • Pla Paskal'
RU2330023C2
NEW BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS MEDICINAL AGENTS 2004
  • Puatu Lidi
  • Bro Valeri
  • Sakjur Karol'
  • Ruber P'Er
  • Pla Paskal'
RU2369601C2
NOVEL DERIVATIVES OF BENZIMIDAZOLE AND THEIR USING AS MEDICAMENTS 2002
  • Puatu Lidi
  • Bro Valeri
  • Ferrandi Ehrik
  • Tjur'O Kristof
RU2294326C2
4-AMINOPIPERIDINE DERIVATIVES, METHODS FOR THEIR PREPARING, COMPOUNDS, PHARMACEUTICAL COMPOSITION 2000
  • Tjur'O Kristof
  • Gonzales Zherom
  • Muane Kristof
RU2266282C2
PYRIMIDOBENZIMIDAZOLE DERIVATIVES AND APPLICATION THEREOF AS AGONISTS OR ANTAGONISTS OF MELANOCORTIN RECEPTORS 2005
  • Puatu Lidi
  • Sakjur Karol'
  • Bro Valeri
  • Ruber P'Er
  • Pla Paskal'
RU2392279C2
5-SULPHANYL-4H-1,2,4-TRIAZOLE DERIVATIVE AND THEIR USE AS MEDICINAL AGENTS 2002
  • Gal'Sera Kontur Mari-Odil'
  • Sidju Al'Ban
  • Ruber P'Er
  • Tjur'O Kristof
RU2367655C2
CONDENSED TRICYCLIC BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY 2014
  • Aleksander Rikki Piter
  • Kalmiano Mark Daniel
  • Defejs Sabine
  • Dyure Veronik
  • Delini Mikhael
  • Kher Yag Paul
  • Dzhekson Viktoriya Elizabet
  • Keje Zhan
  • Kroplin Boris
  • Mak-Koss Malkolm
  • Sabnis Jogesh Anil
  • Selbi Mattyu Dankan
  • Svinnen Dominik Lui Leon
  • Van-Khautvin Natali
  • Chzhu Chzhaonin
  • Vener Folkmar
  • Khajnelt Uve
RU2689777C1
DERIVATIVES OF HYDANTOINS, THIOHYDANTOINS, PYRIMIDINEDIONES AND THIOXOPYRIMIDINEDIONES, METHOD FOR THEIR PREPARING (VARIANTS), INTERMEDIATE COMPOUNDS AND PHARMACEUTICAL COMPOSITION 2000
  • Puatu Lidi
  • Tjur'O Kristof
  • Bro Valeri
RU2277093C2
COMPOUNDS FOR THE TREATMENT OF CERTAIN LEUKOSIS 2019
  • Romero, F. Anthony
  • Kirschberg, Thorsten A.
  • Halcomb, Randall
  • Xu, Yingzi
RU2804709C2
CONDENSED TRICYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY 2014
  • Alekszander Rikki Piter
  • Braun Dzhulien Alister
  • Delini Mikhael
  • Kher Yag Paul
  • Dzhekson Viktoriya Elizabet
  • Yadot Sofie
  • Kroplin Boris
  • Mak-Koss Malkolm
  • Sabnis Jogesh Anil
  • Svinnen Dominik Lui Leon
  • Van-Khautvin Natali
  • Chzhu Chzhaonin
RU2700004C1

RU 2 358 974 C2

Authors

Puatu Lidi

Bro Valeri

Sakjur Karol'

Ruber P'Er

Pla Paskal'

Dates

2009-06-20Published

2004-03-29Filed