5-SULPHANYL-4H-1,2,4-TRIAZOLE DERIVATIVE AND THEIR USE AS MEDICINAL AGENTS Russian patent published in 2009 - IPC C07D249/12 C07D405/04 C07D403/04 C07D409/04 C07D401/04 C07D417/04 C07D403/12 C07D403/14 A61K31/4196 A61P35/00 

Abstract RU 2367655 C2

FIELD: chemistry.

SUBSTANCE: new 5-sulphanyl-4H-1,2,4-triazole derivatives of general formula I (meaning of radicals R1-R3 are indicated in the description of the invention), methods of their preparation by liquid-phase parallel synthesis and pharmaceutical composition are claimed.

EFFECT: claimed compounds display high affinity to some subtypes of somostatin receptors of the SST2 and SST5 subtypes and possibility of their usage for treatment of pathological states or diseases involving one or more of the given somostatin receptors

9 cl, 708 ex

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RU 2 367 655 C2

Authors

Gal'Sera Kontur Mari-Odil'

Sidju Al'Ban

Ruber P'Er

Tjur'O Kristof

Dates

2009-09-20Published

2002-11-27Filed