BENZOXAZINE AND QUINOXALINE DERIVATIVES AND USE THEREOF Russian patent published in 2010 - IPC C07D265/36 C07D413/04 C07D413/06 A61K31/536 A61P25/00 

Abstract RU 2382036 C2

FIELD: chemistry.

SUBSTANCE: described are compounds of formula ; or their pharmaceutically acceptable salts, where A is phenyl, X is CH2- or C=O; Y is O; k equals 1; m equals 0; R2 and R3 each independently represents hydrogen or alkyl, R4 is a group of formula or . Disclosed compounds have selective affinity to 5-HT6 and 5-HT2A receptors. Also described is a pharmaceutical composition containing said compounds and use of the said compounds in making a medicinal agent for treating diseased conditions of the central nervous system.

EFFECT: more effective treatment.

49 cl, 1 tbl, 16 ex

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RU 2 382 036 C2

Authors

Bonkhaus Duglas Vill'Jam

Martin Rene Sharon

Setkhofer Stiven

Chzhan Li

Chzhao Shu-Khaj

Dates

2010-02-20Published

2005-09-22Filed