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(19)

(11)

2 470 022

(13)

(51)

IPC

C07D471/04(2006-01-01)

C07D413/14(2006-01-01)

C07D417/14(2006-01-01)

A61K31/435(2006-01-01)

A61P31/00(2006-01-01)

C07D519/00(2006-01-01)

(21) (22)

Application

2009141311/04, 2008-04-11

(24)

Start date

2008-04-11

(22)

Actual filing date

2008-04-11

(45)

Published

2012-12-20

(72)

Inventor

Bur Daniel'Khubshverlen KristianRjuehdi GeorgSjurive Zhan-FilippTsumbrunn-Aklen Kornelija

(73)

Holder

Aktelion Farmas'Jutiklz Ltd

OXAZOLIDINE ANTIBIOTICS Russian patent published in 2012 - IPC C07D471/04 C07D413/14 C07D417/14 A61K31/435 A61P31/00 C07D519/00

Abstract RU 2470022 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention relates to derivatives of antibiotics, which represent compounds of formula (I) and their pharmaceutically acceptable salts, where U, V, W, X, R¹, R², R³, R⁴, R⁵, R⁶, A, B, D, E, G, m and n are determined in description. Invention also relates to pharmaceutical composition, containing said compounds and their application for obtaining medication for prevention or treatment of bacterial infections.

EFFECT: obtaining useful antimicrobial agents, efficient against various pathogens of people and animals.

23 cl, 1 tbl, 186 ex

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RU 2 470 022 C2

Authors

Bur Daniel'

Khubshverlen Kristian

Rjuehdi Georg

Sjurive Zhan-Filipp

Tsumbrunn-Aklen Kornelija

Dates

2012-12-20—Published

2008-04-11—Filed