PHARMACEUTICAL COMPOSITION OF CARBOXAMIDE INHIBITORS OF HIV INTEGRASE, CONTAINING COMPOSITION WITH CONTROLLED RATE OF RELEASE Russian patent published in 2010 - IPC A61K31/513 A61K9/22 A61P31/18 

Abstract RU 2382648 C2

FIELD: medicine.

SUBSTANCE: invention relates to pharmaceutical composition, suitable for peroral introduction in form of solid medicinal form, which contains efficient amount of main salt of formula compound and composition with controlled rate of release, which contains solubilising agent, gel-forming agent and eater-soluble filler.

EFFECT: compositions are suitable for application in inhibiting of HIV integrase, treatment and prevention of HIV infection, and in treatment, prevention and retardation of AIDS development.

15 cl, 4 dwg, 8 ex

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RU 2 382 648 C2

Authors

Purkavoos Nazaneen

Nej Dzhejms R.

Krjuehjns Marija T.

Vu Jun'Khuehj

Palkar Saurabkh A.

Dates

2010-02-27Published

2005-12-02Filed