1-(3-MORPHOLINOPROPYL)-2-PHENYLIMIDAZO[1,2-a]-BENZIMIDAZOLE DIHYDROCHLORIDE, HAVING PURINE P2Y-RECEPTOR ANTAGONIST PROPERTIES, ANTIAGGREGANT AND ANTITHROMBOTIC ACTIVITY Russian patent published in 2010 - IPC C07D487/04 A61K31/5377 A61K31/4188 A61P7/02 

Abstract RU 2391345 C2

FIELD: chemistry.

SUBSTANCE: invention relates to 1-(3-morpholinopropyl)-2-phenylimidazo[1,2-a]benzimidazole dihydrochloride of formula I:

having purine P2Y1-receptor antagonist properties, antiaggregant and antithrombotic activity.

EFFECT: obtaining a new compound which can be used in medicine for making a medicinal drug for therapy of diseases accompanied by increase in thrombogenic potential of the blood: atherosclerosis, ischemic heart disease, diabetic angiopathy.

1 cl, 5 tbl, 1 ex

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RU 2 391 345 C2

Authors

Spasov Aleksandr Alekseevich

Petrov Vladimir Ivanovich

Anisimova Vera Alekseevna

Minkin Vladimir Isaakovich

Chernikov Maksim Valentinovich

Tolpygin Ivan Evgen'Evich

Dates

2010-06-10Published

2008-07-23Filed