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IPC

C07D487/04(2006-01-01)

A61K31/551(2006-01-01)

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Application

2015108717/04, 2015-03-12

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Start date

2015-03-12

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Actual filing date

2015-03-12

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Published

2016-04-27

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Inventor

Divaeva Ljudmila NikolaevnaKuzmenko Tatjana AndreevnaSpasov Aleksandr AlekseevichMorkovnik Anatolij SavelevichAnisimova Vera AlekseevnaKucherjavenko Aida FatikhovnaSirotenko Viktor Sergeevich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovanija Federalnyj Universitet"Gosudarstvennoe Bjudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Professionalnogo Obrazovanija Gosudarstvennyj Meditsinskij Universitet" Ministerstva Zdravookhranenija Rossijskoj Federatsii

HYDROHALIDES OF 11-PHENOXYETHYL AND 11-BENZYL-SUBSTITUTED 2,3,4,5-TETRAHYDRO[1,3]DIAZEPINO[1,2-a] BENZIMIDAZOLE, HAVING ANTIAGGREGANT ACTIVITY Russian patent published in 2016 - IPC C07D487/04 A61K31/551

Abstract RU 2582618 C1

FIELD: chemistry.

SUBSTANCE: invention relates to hydrogen halides 11 1-(2-phenoxyethyl)-and 11-benzylated 2, 3, 4, 5-tetrahydro [1.3] diazepine [1.2-a] benzimidazole derivatives of formula i: , where R = CH₂OC₆H₄(4-Cl); CH₂OC₂H₄(4-OCH₃); C₆H₄(4-F); X = Cl, Br.

EFFECT: technical outcome is the new derivatives of 2, 3, 4, 5-tetrahydro [1_3] diazepine [1_2-a] benzimidazole derivatives, having antiaggregant activity.

4 cl, 2 tbl, 3 ex

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RU 2 582 618 C1

Authors

Divaeva Ljudmila Nikolaevna

Kuzmenko Tatjana Andreevna

Spasov Aleksandr Alekseevich

Morkovnik Anatolij Savelevich

Anisimova Vera Alekseevna

Kucherjavenko Aida Fatikhovna

Sirotenko Viktor Sergeevich

Dates

2016-04-27—Published

2015-03-12—Filed