FIELD: chemistry.
SUBSTANCE: method of obtaining compound of the formula VIII where R12 and R13 each are removable protective group where protective group R12 is more resistant to extraction by hydrolysis or hydration than R13. Method involves reaction of compound of the formula IX with relevant R12 donor compound selected out of anhydrides, halogenides, carbamates and N-hydroxysuccinimides.
EFFECT: improved method.
4 cl, 6 ex
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Authors
Dates
2010-06-20—Published
2003-12-11—Filed