METHOD OF 4-HYDROXYPROLINE SUBSTRUCTURE-CONTAINING COMPOUND SYNTHESIS Russian patent published in 2010 - IPC C07C227/14 C07D207/16 C07K5/78 

Abstract RU 2392265 C2

FIELD: chemistry.

SUBSTANCE: method of obtaining compound of the formula VIII where R12 and R13 each are removable protective group where protective group R12 is more resistant to extraction by hydrolysis or hydration than R13. Method involves reaction of compound of the formula IX with relevant R12 donor compound selected out of anhydrides, halogenides, carbamates and N-hydroxysuccinimides.

EFFECT: improved method.

4 cl, 6 ex

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Authors

Vitfel'D Bernkhard

Prikoshovikh Val'Ter

Ehrb Bernkhard

Pakhinger Verner

Dates

2010-06-20Published

2003-12-11Filed