COMBINATIONS OF ACTIVATOR (ACTIVATORS) OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR (PPAR), AND INHIBITOR (INHIBITORS) OF STEROL ABSORPTION AND TREATMENT OF VASCULAR DISEASES Russian patent published in 2013 - IPC A61K31/397 A61P9/00 

Abstract RU 2483724 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention relates to field of pharmaceutics and medicine and deals with pharmaceutical composition or therapeutic combination for treatment of vascular pathological states, diabetes, obesity and reduction of concentration of sterols in plasma, which include: (a) at least, one activator of peroxisome proliferator-activated receptor, selected from group, consisting of fenofibrate, clofibrate, gemfibrozil, cyprofibrate, bezafibrate, clinofibrate, binifibrate, lifibrole or their mixture, and (b) sterol absorption inhibitor, represented by formula

, or its pharmaceutically acceptable salt.

EFFECT: claimed are combinations of activator (activators) of peroxisome proliferator-activated receptor (ppar), and inhibitor (inhibitors) of sterol absorption and treatment of vascular diseases.

Similar patents RU2483724C2

Title Year Author Number
APPLICATION OF SUBSTITUTED AZETIDINONES FOR TREATMENT OF SYTOSTEROLEMIA 2002
  • Devis Garri R
RU2756946C2
SUGAR RESIDUE-SUBSTITUTED 2-AZETHIDINONES USEFUL FOR USING AS HYPOCHOLESTEROLEMIC PREPARATIONS 2001
  • Gosal Anima
  • Zbajda Shmuel
  • Chaudkhuri Svaran K.
  • Jannuchi Robert M.
  • Feng Venking
  • Olton Kevin B.
  • Patrik Dzhejms E.
  • Dehjvis Kharri R.
RU2297422C2
COMBINATION OF IAP AND FLT3 INHIBITORS 2007
  • Griffin Dzhejms Duglas
  • Zauehl Li
RU2456983C2
PIPERIDINYLPIPERAZINE DERIVATIVES APPLICABLE AS CHEMOKINE RECEPTOR INHIBITORS 2006
  • Chan Tze-Ming
  • Koks Kehtlin
  • Feng Venking
  • Miller Majkl V.
  • Uehston Dehniehl
  • Makkombi Stjuart V.
RU2411241C2
COMBINED THERAPY INCLUDING SGLT INHIBITORS AND DPP4 INHIBITORS 2009
  • Ueta Kiitiro
  • Arakava Kendzi
  • Matsusita Jasuaki
RU2481106C2
COMBINATIONS WHICH INCLUDE RECEPTOR S1P AGONIST AND JAK3 KINASE INHIBITOR 2005
  • Lejk Filip
RU2415678C2
INHIBITORS OF FACTOR VIIA 2000
  • Klingler Otmar
  • Shudok Manfred
  • Tsoller Gerkhard
  • Khajnel'T Uve
  • Defossa Ehlizabet
  • Matter Khans
  • Safar Pavel
RU2248359C2
NEW INHIBITORS OF 17 β-HYDROXYSTEROID-DEHYDROGENASE TYPE I 2004
  • Messinger Iozef
  • Tole Genrikh-Khubert
  • Khuzen Bettina
  • Van-Stehn Bartolomeus-Jokhannes
  • Shnajder D'Jula
  • Khulsof Jogannes-Bernardus-Ehverardus
  • Koskimies Pasi
  • Jukhansson Nina
  • Adamski Ezhi
RU2369614C2
COMBINATED INHIBITORS OF FBP-ASE AND ANTIDIABETIC AGENTS FOR DIABETES TREATMENT 2001
  • Van Pul'E Paul' D.
  • Ehrion Mark D.
  • Fudzivara Tosikhiko
RU2328308C2
CONJUGATES OF BINDER (ADC) WITH KSP INHIBITORS 2014
  • Lerkhen Khans-Georg
  • Vittrok Sven
  • Gribenov Nils
  • Shtelte-Ludvig Beatriks
  • Zommer Anette
  • Berndt Zandra
  • Malert Kristof
  • Lobell Mario
  • Teryung Karsten
  • Greven Zimone
  • Kancho Grande Iolanda
RU2698697C2

RU 2 483 724 C2

Authors

Kosoglou Teddi

Dehvis Garri R.

Pikar Zhill' Zhan Bernar

Sho Ving-Ki Filip

Dates

2013-06-10Published

2008-11-14Filed