MALIC ACID SALTS AND (3S,5S)-7-[3-AMINO-5-METHYLPIPERIDINYL]-1-CYCLOPROPYL-1,4-DIHYDRO-8-METHOXY-4-OXO-3-CHINOLINE CARBOXYLIC ACID POLYMORPHS Russian patent published in 2011 - IPC C07D401/04 A61K31/4709 A61P31/00 

Abstract RU 2417222 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to (3S,5S)-7-[3-amino-5-methylpiperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-chinoline carboxylic acid malate salts and polymorphs.

EFFECT: invention refers to the pharmaceutical composition containing the described salts and polymorphs which can find application in medicine for treatment or prevention of infectious disorders.

16 cl, 13 dwg, 1 tbl, 9 ex

Similar patents RU2417222C2

Title Year Author Number
INTERMEDIATE COMPOUNDS AND METHODS OF OBTAINING 4-(ACETYLAMINO)-3-[(4-CHLOROPHENYL)THIO]-2-METHYL-1H-INDOLE-1-OF ACETIC ACID 2010
  • Ainge Debra
  • Butters Michael
  • Merifield Eric
  • Ramakrishnan Ravi
  • Rayapati Ravi Naidu
  • Sharma Parhalad Ray
  • Thomson Colin
RU2551852C2
SOLID FORMS (2S,3R,4R,5S,6R)-2-(4-CHLORO-3-(4-ETHOXYBENZIL)PHENYL)-6-(METHYLTHIO)TETRAHYDRO-2H-PYRAN-3,4,5-TRIOL AND METHODS FOR THEIR OBTAINING 2009
  • De Pol' S'Juzan Margaret
  • Perlberg Anett
  • Chzhao Mehtt'Ju Manchzhu
RU2505543C2
METHOD AND PROCESS OF PREPARATION AND PRODUCTION OF DEUTERATED OMEGA-DIPHENYLUREA 2011
  • Fehn Vehjdun
  • Gao Sjaojun
  • Daj Sjaotszjun'
RU2527037C2
SYNTHESIS AND NEW SALINE FORMS OF (R)-5-((E)-2-(PYRROLIDIN-3-YLVINYL)PYRIMIDINE 2009
  • Akireddi Srinivisa Rao
  • Bkhatti Balvinder Singkh
  • Katbertson Timoti Dzh.
  • Dall Gari Moris
  • Miller Krehjg Kharrison
  • Mitchener Ml., Dzhozef Pajk
  • Mun'Os Khulio A.
  • Otten Piter Al'Bert
RU2533819C2
SYNTHESIS AND NOVEL SALT FORMS OF (R)-5-((E)-2-PYRROLIDIN-3-YLVINYL)PYRIMIDINE 2014
  • Akireddi Srinivasa Rao
  • Bkhatti Balvinder Singkh
  • Katbertson Timoti Dzh.
  • Dall Gari Moris
  • Miller Krejg Kharrison
  • Mitchener Ml. Dzhozef Pajk
  • Munos Khulio A.
  • Otten Piter Albert
RU2700796C2
SALT OF OMECAMTIV MECARBIL AND PROCESS FOR PREPARING SAME 2014
  • Tsuj Shen
  • Morrison Genri
  • Nagapudi Kartkhik
  • Uoker Shon
  • Bernard Charlz
  • Khansen Karl Bennett
  • Lanzhill Nil Fred
  • Allgajer Alan Martin
  • Mennen Stiven
  • Vu Zhaklin
  • Morgan Bredli Pol
  • Muchi Aleks
RU2663663C2
TARTRATE 3-((1R,3R)-1-(2,6-DIFLUORINE-4-((1-(3- FLUOROPROPYL)AZETIDINE-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-b]INDOLE-2-YL)-2,2-DIFLUOROPROPANE-1-OL, ITS SOLID FORMS, METHOD OF ITS PREPARATION AND THEIR APPLICATION 2019
  • Chunk, Chol Keun
  • Syuj, Tsze
  • Iding, Khans
  • Klagg, Kajl
  • Delzil, Majkl
  • Fettes, Alek
  • Gosselin, Frensis
  • Lim, Ngiap-Kie
  • Makklori, Endryu
  • Chzhan, Khajmin
  • Chakravarti, Paroma
  • Nagapudi, Kartik
  • Robinson, Sara
RU2809220C2
PROCESS FOR PREPARATION OF N-[(3-AMINOOXETAN-3-YL)METHYL]-2-(1,1-DIOXO-3,5-DIHYDRO-1,4-BENZOTHIAZEPINE-4-YL)-6-METHYL-QUINAZOLINE-4-AMINE 2015
  • Chen Tszyunli
  • Zhen I
  • She Tszin
  • Van Lin
  • Yuj Tszyankhua
  • Chzhan Gotsaj
RU2664643C2
METHODS OF PRODUCING (3R, 3aS, 6aR) HEXAHYDROFURO[2,3-b]FURAN-3-OL 2005
  • Kvadflig Peter Jan Leonard Mario
  • Kestelejn Bart Rudol'F Romani
  • Vejn Robert Jan
  • Libregts Konstantinus Simon Marija
  • Koistra Jakob Khermanus Matteus Khero
  • Lommen Fransiskus Al'Fons Mari
RU2421458C2
METHOD OF PRODUCING (S)-3-HYDROXY-1-(1H-INDOL-5-YL)-2-OXO-PYRROLIDINE-3-CARBOXYLIC ACID 3,5-DIFLUORO-BENZYLAMIDE 2020
  • Heinrich Timo
  • Seenisamy Jeyaprakashnarayanan
RU2826010C2

RU 2 417 222 C2

Authors

Redman-Furij Nansi Li

Godlevski Dzhehjn Ehllen

Diks Majkl Llojd

Dates

2011-04-27Published

2007-03-26Filed