PHARMACEUTICALLY ACCEPTABLE SALTS OF (S)-N-[4-(1-ADAMANTYL)BENZOYL]-α-AMINO ACIDS AND SYNTHESIS METHOD THEREOF Russian patent published in 2011 - IPC C07D233/66 C07D233/64 C07D209/14 C07C233/87 C07C323/29 

Abstract RU 2417988 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds - pharmaceutically acceptable salts of (S)-N-[4-(1-adamantyl)benzoyl]-α-amino acids of general formula (1) , where A+ denotes an ion of an alkali metal, ammonia and N+(C1-4alkyl)4, R2 provided that R1 denotes a hydrogen atom, radicals -CH3, -CH(CH3)2, -CH2CH(CH3)2, -CH(CH3)CH2CH3, CH2-CH2-SH, -CH2-CH2-S-CH3, R1 and R2 together denote a biradical -CH2-CH2-CH2-, closed in the pyrrolidine ring, as well as a method of producing said compounds.

EFFECT: improved method of producing the said compounds.

23 cl, 7 tbl, 1 dwg

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RU 2 417 988 C2

Authors

Krasnikov Sergej Vladislavovich

Ivanova Elena Anatol'Evna

Obukhova Tat'Jana Aleksandrovna

Balakin Konstantin Valer'Evich

Dates

2011-05-10Published

2009-07-02Filed