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(19)

(11)

2 424 237

(13)

(51)

IPC

C07D333/52(2006-01-01)

C07D333/54(2006-01-01)

A61K31/381(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2006131369/04, 2006-08-31

(24)

Start date

2006-08-31

(22)

Actual filing date

2006-08-31

(45)

Published

2011-07-20

(72)

Inventor

Lafaj ZhanRondo BenuaKarniato DeniBonne Pol'Klerk T'ErriShilds ZhaklinDjuk IgorDjuranti Ehrik

(73)

Holder

Laboratuar Terameks

SULPHAMATE DERIVATIVES OF BENZOTHIOPHENE AS STEROID SULPHATASE INHIBITORS Russian patent published in 2011 - IPC C07D333/52 C07D333/54 A61K31/381 A61P35/00

Abstract RU 2424237 C2

FIELD: chemistry.

SUBSTANCE: invention relates to sulphamate derivatives of benzothiophene of formula or

where R₁, R₂, R₃, m and n assume values given in the claim.

EFFECT: possibility of use in treating oestrogen-dependent diseases.

38 cl, 63 ex, 10 tbl

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RU 2 424 237 C2

Authors

Lafaj Zhan

Rondo Benua

Karniato Deni

Bonne Pol'

Klerk T'Erri

Shilds Zhaklin

Djuk Igor

Djuranti Ehrik

Dates

2011-07-20—Published

2006-08-31—Filed