CARBAMOYL BENZOTRIAZOLE DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS Russian patent published in 2011 - IPC C07D249/18 C07D403/12 C07D405/12 C07D409/12 C07D409/14 A61K31/4192 A61P3/00 

Abstract RU 2430096 C2

FIELD: chemistry.

SUBSTANCE: invention describes novel carbamoyl benzotriazole derivatives of general formula , (values of radicals are given in the description), tautomers thereof and pharmaceutically acceptable salts and use thereof as endothelial lipase inhibitors.

EFFECT: improved properties of the derivatives.

11 cl, 148 ex

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RU 2 430 096 C2

Authors

Petri Shtefan

Tsoller Gerkhard

Tennagel'S Norbert

Mjuller Gjunter

Dates

2011-09-27Published

2006-10-12Filed