2-(4-HYDROXY-3-METHOXYPHENYL)-4,7-DIMETHYL-3,4,4a,5,8,8a-HEXAHYDRO-2H-CHROMEN-4,8-DIOL - NOVEL ANALGESIC AGENT Russian patent published in 2011 - IPC C07D311/74 A61K31/352 A61P23/00 

Abstract RU 2430100 C1

FIELD: chemistry.

SUBSTANCE: invention relates to 2-(4-hydroxy-3-methoxyphenyl)-4,7-dimethyl-3,4,4a,5,8,8a-hexahydro-2H-chromen-4,8-diol of formula 1, as well as stereoisomers thereof, including optically active forms, as well as in form of salts with metal cations on the phenol group: Such a compound exhibits analgesic activity and can be used in medicine.

EFFECT: compound of formula 1 has low toxicity and can be obtained from readily available natural compound - α-pinene.

5 ex, 2 tbl

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RU 2 430 100 C1

Authors

Tolstikova Tat'Jana Genrikhovna

Pavlova Alla Viktorovna

Morozova Ekaterina Aleksandrovna

Il'Ina Irina Viktorovna

Ardashov Oleg Vasil'Evich

Korchagina Dina Vladimirovna

Volcho Konstantin Petrovich

Salakhutdinov Nariman Faridovich

Dates

2011-09-27Published

2010-02-24Filed