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(19)

(11)

2 430 921

(13)

(51)

IPC

C07D495/04(2006-01-01)

A61K31/55(2006-01-01)

A61P29/00(2006-01-01)

A61P19/02(2006-01-01)

A61P25/04(2006-01-01)

(21) (22)

Application

2008137533/04, 2007-02-21

(24)

Start date

2007-02-21

(22)

Actual filing date

2007-02-21

(45)

Published

2011-10-10

(72)

Inventor

Bollinger P'EtroPrashad MakhavirRiss BernarDoson-King DzhanetKhistand Peter S.Lju JuganKing DzhonatanShmid VinsanShjurkh Fridrikh

(73)

Holder

Novartis Ag

ORGANIC COMPOUNDS Russian patent published in 2011 - IPC C07D495/04 A61K31/55 A61P29/00 A61P19/02 A61P25/04

Abstract RU 2430921 C2

FIELD: chemistry.

SUBSTANCE: invention relates to an azathiabenzo-azulene derivative of formula I

where R₃ denotes C₁-C₆alkyl, R₄ denotes OH, R₅ denotes halogen and R₆ denotes H or halogen, or a pharmaceutically acceptable salt thereof. The invention also relates to a pharmaceutical composition based on said compounds, having anti-inflammatory or analgesic action.

EFFECT: obtained compounds and pharmaceutical composition can be used to treat arthritis and arthritis-related conditions, and for relieving inflammation and pain associated with acute inflammation of body parts, primarily joints, as a result of injury or as a result of arthritic conditions or other diseased conditions.

17 cl, 8 tbl, 9 ex

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RU 2 430 921 C2

Authors

Bollinger P'Etro

Prashad Makhavir

Riss Bernar

Doson-King Dzhanet

Khistand Peter S.

Lju Jugan

King Dzhonatan

Shmid Vinsan

Shjurkh Fridrikh

Dates

2011-10-10—Published

2007-02-21—Filed